Development of Novel Neurokinin 3 Receptor (NK3R) Selective Agonists with Resistance to Proteolytic Degradation-Reference-Cited by-同舟云学术

Development of Novel Neurokinin 3 Receptor (NK3R) Selective Agonists with Resistance to Proteolytic Degradation

Published:2014-10-07 Issue:20 Volume:57 Page:8646-8651
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Misu Ryosuke¹,Oishi Shinya¹,Yamada Ai¹,Yamamura Takashi²,Matsuda Fuko³,Yamamoto Koki¹,Noguchi Taro¹,Ohno Hiroaki¹,Okamura Hiroaki²,Ohkura Satoshi³,Fujii Nobutaka¹

Affiliation:

1. Graduate School of Pharmaceutical Sciences, Kyoto University, Sakyo-ku, Kyoto 606-8501, Japan

2. Animal Physiology Research Unit, National Institute of Agrobiological Sciences, Tsukuba 305-0901, Japan

3. Graduate School of Bioagricultural Sciences, Nagoya University, Nagoya 464-8601, Japan

Funder

Ministry of Education, Culture, Sports, Science, and Technology

Japan Society for the Promotion of Science

Ministry of Agriculture, Forestry and Fisheries

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm500771w

Reference30 articles.

1. Evidence for Modulation of DoDamine-neuronal Function by Tachykinin NK3Receptor Stimulation in Gerbil Mesencephalic Cell Cultures

2. Tachykinin neurokinin-1 and neurokinin-3 receptor-mediated responses in guinea-pig substantia nigra: an in vitro electrophysiological study

3. The rat isolated portal vein: a preparation sensitive to neurokinins, particularly neurokinin B

4. Neurokinins produce selective venoconstriction via NK-3 receptors in the rat mesenteric vascular bed

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