A Novel Assay Reveals That Weakly Basic Model Compounds Concentrate in Lysosomes to an Extent Greater Than pH-Partitioning Theory Would Predict
Author:
Affiliation:
1. Department of Pharmaceutical Chemistry, The University of Kansas, Lawrence, Kansas 66047
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Pharmaceutical Science,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/mp050043s
Reference31 articles.
1. Intracellular drug sequestration events associated with the emergence of multidrug resistance: a mechanistic review
2. Lysosome membrane permeability: implications for drug delivery
3. Cytoplasmic vacuolation of mouse peritoneal macrophages and the uptake into lysosomes of weakly basic substances.
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