Rational Design of 5‘-Thiourea-Substituted α-Thymidine Analogues as Thymidine Monophosphate Kinase Inhibitors Capable of Inhibiting Mycobacterial Growth-Reference-Cited by-同舟云学术

Rational Design of 5‘-Thiourea-Substituted α-Thymidine Analogues as Thymidine Monophosphate Kinase Inhibitors Capable of Inhibiting Mycobacterial Growth

Published:2007-10-02 Issue:22 Volume:50 Page:5281-5292
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Van Daele Ineke¹,Munier-Lehmann Hélène¹,Froeyen Matheus¹,Balzarini Jan¹,Van Calenbergh Serge¹

Affiliation:

1. Laboratory for Medicinal Chemistry (FFW), University of Gent, Harelbekestraat 72, 9000 Ghent, Belgium, Unité de Chimie Organique, URA CNRS2128, Institut Pasteur, Paris 15, France, and Laboratory for Medicinal Chemistry and Laboratory of Virology and Chemotherapy, Rega Institute for Medical Research, Minderbroedersstraat 10, B-3000 Leuven, Belgium

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0706158

Reference49 articles.

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2. Isoniazid prophylaxis for tuberculosis in HIV infection: a meta-analysis of randomized controlled trials

3. An Outbreak of Tuberculosis with Accelerated Progression among Persons Infected with the Human Immunodeficiency Virus

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