Effects of Altering the Electronics of 2-Methoxyestradiol on Cell Proliferation, on Cytotoxicity in Human Cancer Cell Cultures, and on Tubulin Polymerization-Reference-Cited by-同舟云学术

Effects of Altering the Electronics of 2-Methoxyestradiol on Cell Proliferation, on Cytotoxicity in Human Cancer Cell Cultures, and on Tubulin Polymerization

Published:2004-09-16 Issue:21 Volume:47 Page:5126-5139
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Edsall Allison B.¹,Mohanakrishnan Arasambattu K.¹,Yang Donglai¹,Fanwick Philip E.¹,Hamel Ernest¹,Hanson Arthur D.¹,Agoston Gregory E.¹,Cushman Mark¹

Affiliation:

1. Department of Medicinal Chemistry and Molecular Pharmacology, School of Pharmacy and Pharmacal Sciences, and Department of Chemistry, Purdue University, West Lafayette, Indiana 47907, Screening Technologies Branch, Developmental Therapeutics Program, Division of Cancer Treatment and Diagnosis, National Cancer Institute at Frederick, National Institutes of Health, Frederick, Maryland 21702, and EntreMed, Inc., Rockville, Maryland 20850

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049647a

Reference37 articles.

1. Aromatic Hydroxylation of Estrogens

2. Biogenese von 2-Methoxy-oestradiol-(17?) in der menschlichen Leber

3. The excretion of five different 2-hydroxyoestrogen monomethyl ethers in human pregnancy urine

4. The endogenous oestrogen metabolite 2-methoxyoestradiol inhibits angiogenesis and suppresses tumour growth

5. The cytotoxic effects of estradiol-17β, catecholestradiols and methoxyestradiols on dividing MCF-7 and Hela cells

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