A Click Chemistry Approach to Pleuromutilin Derivatives, Part 2: Conjugates with Acyclic Nucleosides and Their Ribosomal Binding and Antibacterial Activity-Reference-Cited by-同舟云学术

A Click Chemistry Approach to Pleuromutilin Derivatives, Part 2: Conjugates with Acyclic Nucleosides and Their Ribosomal Binding and Antibacterial Activity

Published:2012-02-16 Issue:5 Volume:55 Page:2067-2077
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Dreier Ida¹,Kumar Surender¹,Søndergaard Helle¹,Rasmussen Maria Louise¹,Hansen Lykke Haastrup¹,List Nanna Holmgaard¹,Kongsted Jacob¹,Vester Birte¹,Nielsen Poul¹

Affiliation:

1. Nucleic Acid Center, §Department of Physics, Chemistry and Pharmacy, and ∥Department of Biochemistry and Molecular Biology, University of Southern Denmark, 5230 Odense M, Denmark

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm201266b

Reference26 articles.

1. Antibiotic Substances From Basidiomycetes: VIII. Pleurotus Multilus (Fr.) Sacc. and Pleurotus Passeckerianus Pilat

2. Retapamulin

3. The pleuromutilin drugs tiamulin and valnemulin bind to the RNA at the peptidyl transferase centre on the ribosome

4. Interaction of Pleuromutilin Derivatives with the Ribosomal Peptidyl Transferase Center

5. Inhibition of peptide bond formation by pleuromutilins: the structure of the 50S ribosomal subunit from Deinococcus radiodurans in complex with tiamulin

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