Mechanism of Inactivation of γ-Aminobutyric Acid Aminotransferase by (1S,3S)-3-Amino-4-difluoromethylene-1-cyclopentanoic Acid (CPP-115)-Reference-Cited by-同舟云学术

Mechanism of Inactivation of γ-Aminobutyric Acid Aminotransferase by (1S,3S)-3-Amino-4-difluoromethylene-1-cyclopentanoic Acid (CPP-115)

Published:2015-02-10 Issue:7 Volume:137 Page:2628-2640
ISSN:0002-7863
Container-title:Journal of the American Chemical Society
language:en
Short-container-title:J. Am. Chem. Soc.

Author:

Lee Hyunbeom¹,Doud Emma H.¹²,Wu Rui³,Sanishvili Ruslan⁴,Juncosa Jose I.¹,Liu Dali³,Kelleher Neil L.¹²,Silverman Richard B.¹²

Affiliation:

1. Department of Chemistry, Chemistry of Life Processes Institute, and Center for Molecular Innovation and Drug Discovery, Northwestern University, 2145 Sheridan Road, Evanston, Illinois 60208-3113, United States

2. Department of Molecular Biosciences, Northwestern University, Evanston, Illinois 60208, United States

3. Department of Chemistry and Biochemistry, Loyola University Chicago, 1068 W. Sheridan Road, Chicago, Illinois 60660, United States

4. X-ray Science Division, Argonne National Laboratory, Argonne, Illinois 60439, United States

Funder

National Cancer Institute

National Institute on Drug Abuse

National Institutes of Health

National Institute of General Medical Sciences

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

Link

https://pubs.acs.org/doi/pdf/10.1021/ja512299n

Reference42 articles.

1. Chemical Nature of Synaptic Transmission in Vertebrates

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4. Unrecognized Adult Phenylketonuria

5. Regional activities of metabolic enzymes and glutamate decarboxylase in human brain

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