Selective Inhibition of Human Type-5 17β-Hydroxysteroid Dehydrogenase (AKR1C3) by Baccharin, a Component of Brazilian Propolis-Reference-Cited by-同舟云学术

Selective Inhibition of Human Type-5 17β-Hydroxysteroid Dehydrogenase (AKR1C3) by Baccharin, a Component of Brazilian Propolis

Published:2012-04-16 Issue:4 Volume:75 Page:716-721
ISSN:0163-3864
Container-title:Journal of Natural Products
language:en
Short-container-title:J. Nat. Prod.

Author:

Endo Satoshi¹,Matsunaga Toshiyuki¹,Kanamori Ayano¹,Otsuji Yoko¹,Nagai Hiroko¹,Sundaram Krithika²,El-Kabbani Ossama²,Toyooka Naoki,Ohta Shozo³,Hara Akira¹

Affiliation:

1. Laboratory of Biochemistry, Gifu Pharmaceutical University, Gifu 501-1196, Japan

2. Medicinal Chemistry and Drug Action, Monash Institute of Pharmaceutical Sciences, Parkville, Victoria 3052, Australia

3. Nagaragawa Research Center, API Co., Ltd., Gifu 502-0071, Japan

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Complementary and alternative medicine,Drug Discovery,Pharmaceutical Science,Pharmacology,Molecular Medicine,Analytical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/np201002x

Reference41 articles.

1. Human hydroxysteroid dehydrogenases and pre-receptor regulation: Insights into inhibitor design and evaluation

2. The Aldo-Keto Reductase Superfamily and its Role in Drug Metabolism and Detoxification

3. Carbonyl Reductases and Pluripotent Hydroxysteroid Dehydrogenases of the Short-chain Dehydrogenase/reductase Superfamily

4. Human 3α-hydroxysteroid dehydrogenase isoforms (AKR1C1–AKR1C4) of the aldo-keto reductase superfamily: functional plasticity and tissue distribution reveals roles in the inactivation and formation of male and female sex hormones

Cited by 43 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. AKR1C3 in carcinomas: from multifaceted roles to therapeutic strategies;Frontiers in Pharmacology;2024-03-08

2. Inhibition of aldo-keto reductase 1C3 overcomes gemcitabine/cisplatin resistance in bladder cancer;Chemico-Biological Interactions;2024-01

3. Aldo-Keto Reductase 1C3 Inhibitor Prodrug Improves Pharmacokinetic Profile and Demonstrates In Vivo Efficacy in a Prostate Cancer Xenograft Model;Journal of Medicinal Chemistry;2023-07-10

4. Novel synthetic derivatives of cinnamic and p -coumaric acids with antiproliferative effect on breast MCF-7 tumor cells;Natural Product Research;2023-02-17

5. Artepillin C overcomes apalutamide resistance through blocking androgen signaling in prostate cancer cells;Archives of Biochemistry and Biophysics;2023-02