Discovery of Novel, Potent Benzamide Inhibitors of 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD1) Exhibiting Oral Activity in an Enzyme Inhibition ex Vivo Model▽-Reference-Cited by-同舟云学术

Discovery of Novel, Potent Benzamide Inhibitors of 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD1) Exhibiting Oral Activity in an Enzyme Inhibition ex Vivo Model▽

Published:2008-07 Issue:13 Volume:51 Page:3953-3960
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Julian Lisa D.,Wang Zhulun,Bostick Tracy,Caille Seb,Choi Rebekah,DeGraffenreid Michael,Di Yongmei,He Xiao,Hungate Randall W.,Jaen Juan C.,Liu Jinsong,Monshouwer Mario,McMinn Dustin,Rew Yosup,Sudom Athena,Sun Daqing,Tu Hua,Ursu Stefania,Walker Nigel,Yan Xuelei,Ye Qiuping,Powers Jay P.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm800310g

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