A Potent, Nonpeptidyl 1H-Quinolone Antagonist for the Gonadotropin-Releasing Hormone Receptor-Reference-Cited by-同舟云学术

A Potent, Nonpeptidyl 1H-Quinolone Antagonist for the Gonadotropin-Releasing Hormone Receptor

Published:2001-03-01 Issue:6 Volume:44 Page:917-922
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

DeVita Robert J.¹,Walsh Thomas F.¹,Young Jonathan R.¹,Jiang Jinlong¹,Ujjainwalla Feroze¹,Toupence Richard B.¹,Parikh Mamta¹,Huang Song X.¹,Fair Jason A.¹,Goulet Mark T.¹,Wyvratt Matthew J.¹,Lo Jane-L.¹,Ren Ning¹,Yudkovitz Joel B.¹,Yang Yi T.¹,Cheng Kang¹,Cui Jisong¹,Mount George¹,Rohrer Susan P.¹,Schaeffer James M.¹,Rhodes Linda¹,Drisko Jennifer E.¹,McGowan Erin¹,MacIntyre D. Euan¹,Vincent Styliani¹,Carlin Josephine R.¹,Cameron Judith¹,Smith Roy G.¹

Affiliation:

1. Departments of Medicinal Chemistry, Biochemistry & Physiology, Pharmacology, and Drug Metabolism, Merck Research Laboratories, P.O. Box 2000, Rahway, New Jersey 07065-0900, and Oregon Regional Primate Research Center, Oregon Health Sciences University, 505 NW 185th Avenue, Beaverton, Oregon 97006

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm000275p

Reference13 articles.

1. Structure of the porcine LH- and FSH-releasing hormone. I. The proposed amino acid sequence

2. Structure of the porcine LH- and FSH-releasing hormone. II. Confirmation of the proposed structure by conventional sequential analyses

3. Conn, P. M.; Janovick, J. A.; Stanislaus, D.; Kuphal, D.; Jennes, L. InVitaminsand Hormones; Litwack, G., Ed.; Academic Press: New York, 1995; Vol. 50, pp 151−214.

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