Design, Synthesis, and Biological Activity of Novel 5-((Arylfuran/1H-pyrrol-2-yl)methylene)-2-thioxo-3-(3-(trifluoromethyl)phenyl)thiazolidin-4-ones as HIV-1 Fusion Inhibitors Targeting gp41-Reference-Cited by-同舟云学术

Design, Synthesis, and Biological Activity of Novel 5-((Arylfuran/1H-pyrrol-2-yl)methylene)-2-thioxo-3-(3-(trifluoromethyl)phenyl)thiazolidin-4-ones as HIV-1 Fusion Inhibitors Targeting gp41

Published:2010-12-29 Issue:2 Volume:54 Page:572-579
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Jiang Shibo¹,Tala Srinivasa R.²,Lu Hong¹,Abo-Dya Nader E.²³,Avan Ilker²⁴,Gyanda Kapil²,Lu Lu¹,Katritzky Alan R.²,Debnath Asim K.¹

Affiliation:

1. Lindsley F. Kimball Research Institute, New York Blood Center, New York 10065, United States

2. Center for Heterocyclic Compounds, Department of Chemistry, University of Florida, Gainesville, Florida 32611, United States

3. Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Zagazig University, Zagazig, 44519, Egypt

4. Department of Chemistry, Anadolu University, 26470, Eskişehir, Turkey

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm101014v

Reference39 articles.

1. The prevalence of antiretroviral drug resistance in the United States

2. Adverse effects of antiretroviral therapy

3. Mechanisms of Viral Membrane Fusion and Its Inhibition

4. The entry of entry inhibitors: A fusion of science and medicine

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