An Efficient and Expeditious Synthesis of Di- and Trisubstituted Amino-phenyl and -benzyl Derivatives of Tetrazole and [1,3,4]Oxadiazol-2-one-Reference-Cited by-同舟云学术

An Efficient and Expeditious Synthesis of Di- and Trisubstituted Amino-phenyl and -benzyl Derivatives of Tetrazole and [1,3,4]Oxadiazol-2-one

Published:2008-08-16 Issue:5 Volume:10 Page:671-680
ISSN:1520-4766
Container-title:Journal of Combinatorial Chemistry
language:en
Short-container-title:J. Comb. Chem.

Author:

Desforges Gwenaelle¹,Bombrun Agnes¹,Quattropani Anna¹

Affiliation:

1. Merck Serono Geneva Research Center, 9 Chemin des Mines, CH-1202 Geneva, Switzerland, Department of Organic Chemistry, University of Geneva, 30 quai Ernest Ansermet, CH-1211 Geneva 4, Switzerland.

Publisher

American Chemical Society (ACS)

Subject

General Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/cc800083h

Reference28 articles.

1. Bioisosterism: A Useful Strategy for Molecular Modification and Drug Design

2. Bioisosterism: A Rational Approach in Drug Design

3. 5-Substituted-1H-tetrazoles as carboxylic acid isosteres: medicinal chemistry and synthetic methods

4. A new class of angiotensin II receptor antagonists with a novel acidic bioisostere

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