Diastereoselective Synthesis of 2-Phenyl-3-(trifluoromethyl)piperazines as Building Blocks for Drug Discovery-Reference-Cited by-同舟云学术

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Diastereoselective Synthesis of 2-Phenyl-3-(trifluoromethyl)piperazines as Building Blocks for Drug Discovery

Published:2014-06-03 Issue:12 Volume:79 Page:5887-5894
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Sánchez-Roselló María¹,Delgado Oscar²,Mateu Natalia¹,Trabanco Andrés A.²,Van Gool Michiel²,Fustero Santos¹³

Affiliation:

1. Laboratorio de Moléculas Orgánicas, Centro de Investigación Príncipe Felipe, E-46012 Valencia, Spain

2. Neuroscience Medicinal Chemistry Department, Janssen Research and Development, E-45007 Toledo, Spain

3. Departamento de Química Orgánica, Universidad de Valencia, E-46100 Burjassot, Spain

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/jo500832j

Reference52 articles.

1. Methods for drug discovery: development of potent, selective, orally effective cholecystokinin antagonists

2. The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures

3. Privileged scaffolds for library design and drug discovery

4. Characteristic Physical Properties and Structural Fragments of Marketed Oral Drugs

5. DrugBank: a knowledgebase for drugs, drug actions and drug targets

Cited by 21 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Development of a Safe and Practical Synthesis of Enantiomerically Pure (S)- and (R)-N-Boc-3-(Trifluoromethyl)piperazines Enabled by Aza-Michael Addition of Optically Pure 4-Phenyl-2-Oxazolidinone to 3,3,3-Trifluoro-1-Nitropropene;Organic Process Research & Development;2024-07-30

2. Fluorinated Imines in Tandem and Cycloaddition Reactions;The Chemical Record;2023-01-12

3. Phenylglycinol Derived Chemistry;Reference Module in Chemistry, Molecular Sciences and Chemical Engineering;2023

4. A Concise Synthetic Method for Constructing 3-Substituted Piperazine-2-Acetic Acid Esters from 1,2-Diamines;Molecules;2022-05-25

5. Diastereoselective Synthesis of Enantioenriched Trifluoromethylated Ethylenediamines and Isoindolines Containing Two Stereogenic Carbon Centers by Nucleophilic Trifluoromethylation Using HFC-23;The Journal of Organic Chemistry;2020-05-18

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