Dipeptide Boronic Acid Inhibitors of Dipeptidyl Peptidase IV: Determinants of Potency and in Vivo Efficacy and Safety-Reference-Cited by-同舟云学术

Dipeptide Boronic Acid Inhibitors of Dipeptidyl Peptidase IV: Determinants of Potency and in Vivo Efficacy and Safety

Published:2008-09-11 Issue:19 Volume:51 Page:6005-6013
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Connolly Beth A.¹,Sanford David G.¹,Chiluwal Amrita K.¹,Healey Sarah E.¹,Peters Diane E.¹,Dimare Matthew T.¹,Wu Wengen¹,Liu Yuxin¹,Maw Hlaing¹,Zhou Yuhong¹,Li Youhua¹,Jin Zhiping¹,Sudmeier James L.¹,Lai Jack H.¹,Bachovchin William W.¹

Affiliation:

1. Department of Biochemistry, Tufts University, 136 Harrison Avenue, Boston, Massachusetts 02111

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm800390n

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2. Catalytic properties and inhibition of proline-specific dipeptidyl peptidases II, IV and VII

3. Therapeutic potential of dipeptidyl peptidase IV inhibitors for the treatment of type 2 diabetes

4. Degradation of glucose-dependent insulinotropic polypeptide and truncated glucagon-like peptide 1 in vitro and in vivo by dipeptidyl peptidase IV.

5. Investigation of Glucose-dependent Insulinotropic Polypeptide(1-42) and Glucagon-like Peptide-1-(7-36) Degradation by Dipeptidyl Peptidase IV Using Matrix-assisted Laser Desorption/Ionization-Time of Flight Mass Spectrometry

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