Lipid-Dependent Activation of the Orphan G Protein-Coupled Receptor, GPR3-Reference-Cited by-同舟云学术

Lipid-Dependent Activation of the Orphan G Protein-Coupled Receptor, GPR3

Published:2024-02-20 Issue:5 Volume:63 Page:625-631
ISSN:0006-2960
Container-title:Biochemistry
language:en
Short-container-title:Biochemistry

Author:

Russell Isabella C.¹²,Zhang Xin¹²,Bumbak Fabian¹²^ORCID,McNeill Samantha M.¹,Josephs Tracy M.¹²^ORCID,Leeming Michael G.³,Christopoulos George¹,Venugopal Hariprasad⁴,Flocco Maria M.⁵,Sexton Patrick M.¹²^ORCID,Wootten Denise¹²^ORCID,Belousoff Matthew J.¹²^ORCID

Affiliation:

1. Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville 3052, Victoria Australia

2. Australian Research Council Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville 3052, Victoria Australia

3. Bio21 Molecular Science & Biotechnology Institute, Melbourne Mass Spectrometry and Proteomics Facility, The University of Melbourne, Melbourne, VIC 3052, Australia

4. Ramaciotti Centre for Cryo Electron Microscopy, Monash University, Clayton 3800, Victoria Australia

5. Mechanistic and Structural Biology, Discovery Sciences, BioPharmaceuticals R&D, AstraZeneca, Cambridge CB20AA, United Kingdom

Funder

National Health and Medical Research Council

Australian Research Council

Publisher

American Chemical Society (ACS)

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.biochem.3c00647

Reference19 articles.

1. G Protein-Coupled Receptors as Targets for Approved Drugs: How Many Targets and How Many Drugs?

2. Lipolysis drives expression of the constitutively active receptor GPR3 to induce adipose thermogenesis

3. Common activation mechanism of class A GPCRs

4. G protein–biased GPR3 signaling ameliorates amyloid pathology in a preclinical Alzheimer’s disease mouse model

5. Generation of mouse oocytes defective in cAMP synthesis and degradation: Endogenous cyclic AMP is essential for meiotic arrest

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1. Application of FRET- and BRET-based live-cell biosensors in deorphanization and ligand discovery studies on orphan G protein-coupled receptors;SLAS Discovery;2024-09

2. Shifting our perspective on orphan G protein-coupled receptors;Nature Structural & Molecular Biology;2024-04