Structure of Estradiol Metal Chelate and Estrogen Receptor Complex: The Basis for Designing a New Class of Selective Estrogen Receptor Modulators-Reference-Cited by-同舟云学术

Structure of Estradiol Metal Chelate and Estrogen Receptor Complex: The Basis for Designing a New Class of Selective Estrogen Receptor Modulators

Published:2011-04-19 Issue:10 Volume:54 Page:3575-3580
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Li Min-Jun¹,Greenblatt Harry M.¹,Dym Orly¹,Albeck Shira¹,Pais Adi¹,Gunanathan Chidambaram¹,Milstein David¹,Degani Hadassa¹,Sussman Joel L.¹

Affiliation:

1. Department of Structural Biology, ‡Department of Biological Regulation, §Israel Structural Proteomics Center (ISPC), and ∥Department of Organic Chemistry, Weizmann Institute of Science, Rehovot 76100, Israel

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm200192y

Reference36 articles.

1. Estrogen receptors and human disease

2. Estrogen Receptors: How Do They Signal and What Are Their Targets

3. Capitalizing on the Complexities of Estrogen Receptor Pharmacology in the Quest for the Perfect SERM

4. Preclinical and Clinical Studies on the Use of Platinum Complexes for Breast Cancer Treatment

5. Water-Soluble Contrast Agents Targeted at the Estrogen Receptor for Molecular Magnetic Resonance Imaging

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