4-(Phenylsulfonyl)piperidines: Novel, Selective, and Bioavailable 5-HT2A Receptor Antagonists-Reference-Cited by-同舟云学术

4-(Phenylsulfonyl)piperidines: Novel, Selective, and Bioavailable 5-HT2A Receptor Antagonists

Published:2001-12-20 Issue:2 Volume:45 Page:492-503
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Fletcher Stephen R.¹,Burkamp Frank¹,Blurton Peter¹,Cheng Susan K. F.¹,Clarkson Robert¹,O'Connor Desmond¹,Spinks Daniel¹,Tudge Matthew¹,van Niel Monique B.¹,Patel Smita¹,Chapman Kerry¹,Marwood Rose¹,Shepheard Sara¹,Bentley Graham¹,Cook Gina P¹,Bristow Linda J¹,Castro Jose L.¹,Hutson Peter H.¹,MacLeod Angus M.¹

Affiliation:

1. Merck Sharp and Dohme, The Neuroscience Research Centre, Terlings Park, Eastwick Road, Harlow, Essex CM20 2QR, U.K.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm011030v

Reference32 articles.

1. Section Review Central & Peripheral Nervous Systems: Mirtazapine - a novel antidepressant compound currently undergoing clinical evaluation

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