Crystallographic Fragment Screening and Structure-Based Optimization Yields a New Class of Influenza Endonuclease Inhibitors-Reference-Cited by-同舟云学术

Crystallographic Fragment Screening and Structure-Based Optimization Yields a New Class of Influenza Endonuclease Inhibitors

Published:2013-09-13 Issue:11 Volume:8 Page:2501-2508
ISSN:1554-8929
Container-title:ACS Chemical Biology
language:en
Short-container-title:ACS Chem. Biol.

Author:

Bauman Joseph D.,Patel Disha,Baker Steven F.¹,Vijayan R. S. K.,Xiang Amy²,Parhi Ajit K.²,Martínez-Sobrido Luis¹,LaVoie Edmond J.,Das Kalyan,Arnold Eddy

Affiliation:

1. Department of Microbiology and Immunology, University of Rochester, Rochester, New York 14642, United States

2. TAXIS Pharmaceuticals Inc., North Brunswick, New Jersey 08902, United States

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/cb400400j

Reference51 articles.

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2. CDC (2013) Interim adjusted estimates of seasonal Influenza vaccine effectiveness – United States February 2013. Centers for disease control and prevention. [Online] Availablehttp://www.cdc.gov/mmwr/preview/mmwrhtml/mm6207a2.htm?s_cid= mm6207a2_w.

3. Structures of influenza A proteins and insights into antiviral drug targets

4. Avian influenza A (H5N1) infection: targets and strategies for chemotherapeutic intervention

5. Combination Chemotherapy for Influenza

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