Design, Synthesis, and Evaluation of Proline and Pyrrolidine Based Melanocortin Receptor Agonists. A Conformationally Restricted Dipeptide Mimic Approach-Reference-Cited by-同舟云学术

Design, Synthesis, and Evaluation of Proline and Pyrrolidine Based Melanocortin Receptor Agonists. A Conformationally Restricted Dipeptide Mimic Approach

Published:2006-06-24 Issue:15 Volume:49 Page:4745-4761
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Tian Xinrong¹,Field Timothy B.¹,Switzer Adrian G.¹,Mazur Adam W.¹,Ebetino Frank H.¹,Wos John A.¹,Berberich Steve M.¹,Jayasinghe Lalith R.¹,Obringer Cindy M.¹,Dowty Martin E.¹,Pinney Beth B.¹,Farmer Julie A.¹,Crossdoersen Doreen¹,Sheldon Russell J.¹

Affiliation:

1. Procter & Gamble Pharmaceuticals, Health Care Research Center, 8700 Mason-Montgomery Road, Mason, Ohio 45040

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm060384p

Reference53 articles.

1. Structure and Biosynthesis of Pro-Adrenocorticotropin/Endorphin and Related Peptides*

2. .alpha.-Melanotropin: the minimal active sequence in the frog skin bioassay

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