Industrial Synthesis of the Key Precursor in the Synthesis of the Anti-Influenza Drug Oseltamivir Phosphate (Ro 64-0796/002, GS-4104-02): Ethyl (3R,4S,5S)-4,5-epoxy-3-(1-ethyl-propoxy)-cyclohex-1-ene-1-carboxylate-Reference-Cited by-同舟云学术

Industrial Synthesis of the Key Precursor in the Synthesis of the Anti-Influenza Drug Oseltamivir Phosphate (Ro 64-0796/002, GS-4104-02): Ethyl (3R,4S,5S)-4,5-epoxy-3-(1-ethyl-propoxy)-cyclohex-1-ene-1-carboxylate

Published:1999-06-30 Issue:4 Volume:3 Page:266-274
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Federspiel Muriel¹,Fischer Rolf¹,Hennig Michael¹,Mair Hans-Jürgen¹,Oberhauser Thomas¹,Rimmler Gösta¹,Albiez Thomas¹,Bruhin Jürg¹,Estermann Heinrich¹,Gandert Carsten¹,Göckel Volker¹,Götzö Stephan¹,Hoffmann Ursula¹,Huber Gabriel¹,Janatsch Günter¹,Lauper Stephan¹,Röckel-Stäbler Odette¹,Trussardi Rene¹,Zwahlen Andreas G.¹

Affiliation:

1. F. Hoffmann-La Roche Ltd., CH-4070 Basel, Switzerland

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op9900176

Reference28 articles.

1. Structure−Activity Relationship Studies of Novel Carbocyclic Influenza Neuraminidase Inhibitors

2. Influenza Neuraminidase Inhibitors Possessing a Novel Hydrophobic Interaction in the Enzyme Active Site: Design, Synthesis, and Structural Analysis of Carbocyclic Sialic Acid Analogues with Potent Anti-Influenza Activity

3. Practical Total Synthesis of the Anti-Influenza Drug GS-4104