Identification of a Potent Sodium Hydrogen Exchanger Isoform 1 (NHE1) Inhibitor with a Suitable Profile for Chronic Dosing and Demonstrated Cardioprotective Effects in a Preclinical Model of Myocardial Infarction in the Rat

Author:

Huber John D.1,Bentzien Jörg1,Boyer Stephen J.1,Burke Jennifer1,De Lombaert Stéphane1,Eickmeier Christian2,Guo Xin1,Haist James V.3,Hickey Eugene R.1,Kaplita Paul4,Karmazyn Morris3,Kemper Raymond5,Kennedy Charles A.1,Kirrane Thomas1,Madwed Jeffrey B.6,Mainolfi Elizabeth6,Nagaraja Nelamangara4,Soleymanzadeh Fariba1,Swinamer Alan1,Eldrup Anne B.1

Affiliation:

1. Department of Medicinal Chemistry, Boehringer Ingelheim Pharmaceuticals, Ridgefield, Connecticut 06877, United States

2. Department of Medicinal Chemistry, Boehringer Ingelheim Pharma GmbH & Co KG, 88397 Biberach an der Riss, Germany

3. Department of Physiology & Pharmacology, University of Western Ontario, Medical Sciences Building, London, Ontario N6A 5C1,Canada

4. Drug Discovery Support, Boehringer Ingelheim Pharmaceuticals, Ridgefield, Connecticut 06877, United States

5. Non-Clinical Drug Safety, Boehringer Ingelheim Pharmaceuticals, Ridgefield, Connecticut 06877, United States

6. Cardiometabolic-Disease Research, Boehringer Ingelheim Pharmaceuticals, Ridgefield, Connecticut 06877, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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