Facile Reductive Amination of Aldehydes with Electron-Deficient Anilines by Acyloxyborohydrides in TFA: Application to a Diazaindoline Scale-Up-Reference-Cited by-同舟云学术

Facile Reductive Amination of Aldehydes with Electron-Deficient Anilines by Acyloxyborohydrides in TFA: Application to a Diazaindoline Scale-Up

Published:2009-04-07 Issue:9 Volume:74 Page:3587-3590
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Boros Eric E.¹,Thompson James B.¹,Katamreddy Subba R.¹,Carpenter Andrew J.¹

Affiliation:

1. GlaxoSmithKline Research & Development, Five Moore Drive, Research Triangle Park, North Carolina 27709

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/jo900157z

Reference15 articles.

1. Katamreddy, S. R.; Caldwell, R. D.; Heyer, D.; Samano, V.; Thompson, J. B.; Carpenter, A. J.; Conlee, C. R.; Boros, E. E.; Thompson, B. D.Patent WO 2008/008887 A2;

2. For recent reviews of GPR119 receptor agonists, see:

3. GPR119: “Double-Dipping” for Better Glycemic Control

4. GPR119 agonists as potential new oral agents for the treatment of type 2 diabetes and obesity

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