Synthesis and Biological Activity of a Novel Methylamine-Bridged Enkephalin Analogue (MABE): A New Route to Cyclic Peptides and Peptidomimetics-Reference-Cited by-同舟云学术

Synthesis and Biological Activity of a Novel Methylamine-Bridged Enkephalin Analogue (MABE): A New Route to Cyclic Peptides and Peptidomimetics

Published:1998-06-16 Issue:14 Volume:41 Page:2631-2635
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Shreder Kevin¹,Zhang Li¹,Dang Trunghau¹,Yaksh Tony L.¹,Umeno Hiroshi¹,DeHaven Robert¹,Daubert Jeffrey¹,Goodman Murray¹

Affiliation:

1. Department of Chemistry and Biochemistry, 9500 Gilman Drive, University of California at San Diego, La Jolla, California 92093-0343, Department of Anesthesiology, 9500 Gilman Drive, University of California at San Diego, La Jolla, California 92093-0818, and Adolor Corporation, 395 Pheonixville Pike, Malvern, Pennsylvania 19355

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm970861r

Reference20 articles.

1. Isolation of an endogenous compound from the brain with pharmacological properties similar to morphine

2. Endogenous opiates: 1995

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4. Recent developments in the design of receptor specific opioid peptides

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