The Discovery of Setileuton, a Potent and Selective 5-Lipoxygenase Inhibitor-Reference-Cited by-同舟云学术

The Discovery of Setileuton, a Potent and Selective 5-Lipoxygenase Inhibitor

Published:2010-04-13 Issue:4 Volume:1 Page:170-174
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Ducharme Yves¹,Blouin Marc¹,Brideau Christine¹,Châteauneuf Anne¹,Gareau Yves¹,Grimm Erich L.¹,Juteau Hélène¹,Laliberté Sébastien¹,MacKay Bruce¹,Massé Frédéric¹,Ouellet Marc¹,Salem Myriam¹,Styhler Angela¹,Friesen Richard W.¹

Affiliation:

1. Merck Frosst Centre for Therapeutic Research, 16711 Trans Canada Highway, Kirkland, Quebec, Canada H9H 3L1

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml100029k

Reference18 articles.

1. Leukotrienes

2. 5-Lipoxygenase: regulation of expression and enzyme activity

3. What's all the FLAP about?: 5-lipoxygenase-activating protein inhibitors for inflammatory diseases

4. Therapeutic options for 5-lipoxygenase inhibitors

5. Asthma

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