Studies Examining the Relationship between the Chemical Structure of Protoxin II and Its Activity on Voltage Gated Sodium Channels
Author:
Affiliation:
1. Discovery Research, Purdue Pharma L.P., 6 Cedar Brook Drive, Cranbury, New Jersey 08512, United States
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm500687u
Reference37 articles.
1. Overview of Molecular Relationships in the Voltage-Gated Ion Channel Superfamily
2. Familial pain syndromes from mutations of the Nav1.7 sodium channel
3. Nociceptor-specific gene deletion reveals a major role for Nav1.7 (PN1) in acute and inflammatory pain
4. An SCN9A channelopathy causes congenital inability to experience pain
5. Voltage sensor interaction site for selective small molecule inhibitors of voltage-gated sodium channels
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