Probes for Narcotic Receptor Mediated Phenomena. 34. Synthesis and Structure−Activity Relationships of a Potent μ-Agonist δ-Antagonist and an Exceedingly Potent Antinociceptive in the Enantiomeric C9-Substituted 5-(3-Hydroxyphenyl)-N-phenylethylmorphan Series-Reference-Cited by-同舟云学术

Probes for Narcotic Receptor Mediated Phenomena. 34. Synthesis and Structure−Activity Relationships of a Potent μ-Agonist δ-Antagonist and an Exceedingly Potent Antinociceptive in the Enantiomeric C9-Substituted 5-(3-Hydroxyphenyl)-N-phenylethylmorphan Series

Published:2007-07-11 Issue:16 Volume:50 Page:3765-3776
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Hiebel Anne-Cécile¹,Lee Yong Sok¹,Bilsky Edward¹,Giuvelis Denise¹,Deschamps Jeffrey R.¹,Parrish Damon A.¹,Aceto Mario D.¹,May Everette L.¹,Harris Louis S.¹,Coop Andrew¹,Dersch Christina M.¹,Partilla John S.¹,Rothman Richard B.¹,Cheng Kejun¹,Jacobson Arthur E.¹,Rice Kenner C.¹

Affiliation:

1. Drug Design and Synthesis Section, Chemical Biology Research Branch, National Institute on Drug Abuse, and Center for Molecular Modeling, Division of Computational Bioscience, Center for Information Technology, National Institutes of Health, DHHS, Bethesda, MD 20892, University of New England, College of Osteopathic Medicine, Biddeford, ME 04005, Laboratory for the Structure of Matter, Naval Research Laboratory, Washington, DC 20375, Department of Pharmacology and Toxicology, School of Medicine, Virginia...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm061325e

Reference39 articles.

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