Synthesis of Small 3-Fluoro- and 3,3-Difluoropyrrolidines Using Azomethine Ylide Chemistry-Reference-Cited by-同舟云学术

Synthesis of Small 3-Fluoro- and 3,3-Difluoropyrrolidines Using Azomethine Ylide Chemistry

Published:2015-06-24 Issue:14 Volume:80 Page:7266-7274
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

McAlpine Indrawan¹,Tran-Dubé Michelle¹,Wang Fen¹,Scales Stephanie¹,Matthews Jean¹,Collins Michael R.¹,Nair Sajiv K.¹,Nguyen Mary¹,Bian Jianwei²,Alsina Luis Martinez²,Sun Jianmin²,Zhong Jiaying²,Warmus Joseph S.²,O’Neill Brian T.²

Affiliation:

1. Pfizer Worldwide Medicinal Chemistry, Pfizer Research & Development, 10770 Science Center Drive, San Diego, California 92121, United States

2. Pfizer Worldwide Medicinal Chemistry, Pfizer Research & Development, 445 Eastern Point Road, Groton, Connecticut 06340, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.joc.5b00853

Reference26 articles.

1. The Many Roles for Fluorine in Medicinal Chemistry

2. Predicting and Tuning Physicochemical Properties in Lead Optimization: Amine Basicities

3. Good Partnership between Sulfur and Fluorine: Sulfur-Based Fluorination and Fluoroalkylation Reagents for Organic Synthesis

4. Aminodifluorosulfinium Salts: Selective Fluorination Reagents with Enhanced Thermal Stability and Ease of Handling,

5. Aminodifluorosulfinium Tetrafluoroborate Salts as Stable and Crystalline Deoxofluorinating Reagents

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