Rhodium(III)-Catalyzed C–H Functionalization of 1-(2H)-Phthalazinones at C8
Author:
Affiliation:
1. Discovery Chemistry, Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.joc.6b02522
Reference50 articles.
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2. Vogelsang, D.; Scheffler, G.; Brock, N.; Lenke, D.Basically substituted benzyl phthalazone derivatives, acid salts thereof and process for the production thereof.US Patent 3813384, 1974.
3. 4-[3-(4-Cyclopropanecarbonylpiperazine-1-carbonyl)-4-fluorobenzyl]-2H-phthalazin-1-one: A Novel Bioavailable Inhibitor of Poly(ADP-ribose) Polymerase-1
4. Removable Directing Groups in Organic Synthesis and Catalysis
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