A Protocol for the Synthesis of CF2H-Containing Pyrazolo[1,5-c]quinazolines from 3-Ylideneoxindoles and in Situ Generated CF2HCHN2-Reference-Cited by-同舟云学术

A Protocol for the Synthesis of CF2H-Containing Pyrazolo[1,5-c]quinazolines from 3-Ylideneoxindoles and in Situ Generated CF2HCHN2

Published:2018-06-04 Issue:12 Volume:83 Page:6556-6565
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Han Wen-Yong¹^ORCID,Wang Jian-Shu¹,Zhao Jia¹,Long Lin¹,Cui Bao-Dong¹,Wan Nan-Wei¹,Chen Yong-Zheng¹

Affiliation:

1. Generic Drug Research Center of Guizhou Province, Green Pharmaceuticals Engineering Research Center of Guizhou Province, School of Pharmacy, Zunyi Medical University, Zunyi 563000, China

Funder

National Natural Science Foundation of China

the Science and Technology Department of Guizhou Province

Program for the Top Talents of Science and Technology in Higher Learning Institutions of Guizhou Province

the Fifth Batch of Talent Base in Guizhou Province

National First-Rate Construction Discipline of Pharmacy

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.joc.8b00866

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5. Fluorination methods in drug discovery

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