Salt Selection and Simultaneous Polymorphism Assessment via High-Throughput Crystallization: The Case of Sertraline-Reference-Cited by-同舟云学术

Salt Selection and Simultaneous Polymorphism Assessment via High-Throughput Crystallization: The Case of Sertraline

Published:2003-10-14 Issue:6 Volume:7 Page:990-996
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Remenar Julius F.¹,MacPhee J. Michael¹,Larson Bridget K.¹,Tyagi Viraj A.¹,Ho Jason H.¹,McIlroy David A.¹,Hickey Magali B.¹,Shaw Paul B.¹,Almarsson Örn¹

Affiliation:

1. Transform Pharmaceuticals, Inc., 29 Hartwell Avenue, Lexington, Massachusetts 02421-3102, U.S.A.

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op034115%2B

Reference15 articles.

1. Pharmaceutical Salts

2. Salt selection for basic drugs

3. Bernstein, J. Polymorphism and Patents; InPolymorphism inMolecular Crystals; Oxford: New York, 2002; pp 297−307.

4. An integrated approach to the selection of optimal salt form for a new drug candidate

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