The Structure−Activity Relationship of the Antimalarial Ozonide Arterolane (OZ277)

Author:

Dong Yuxiang1,Wittlin Sergio2,Sriraghavan Kamaraj1,Chollet Jacques2,Charman Susan A.3,Charman William N.3,Scheurer Christian2,Urwyler Heinrich4,Santo Tomas Josefina3,Snyder Christopher2,Creek Darren J.3,Morizzi Julia3,Koltun Maria3,Matile Hugues5,Wang Xiaofang1,Padmanilayam Maniyan1,Tang Yuanqing1,Dorn Arnulf5,Brun Reto2,Vennerstrom Jonathan L.1

Affiliation:

1. College of Pharmacy, University of Nebraska Medical Center, 986025 Nebraska Medical Center, Omaha, NE

2. Swiss Tropical Institute, Socinstrasse 57, CH-4002 Basel, Switzerland

3. Centre for Drug Candidate Optimisation, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), 381 Royal Parade, Parkville, Victoria 3052, Australia

4. Basilea Pharmaceutica Ltd., Grenzacherstrasse 487, CH-4058 Basel, Switzerland

5. F. Hoffmann-La Roche Ltd., Grenzacherstrasse 124, CH-4070 Basel, Switzerland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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