Synthesis and Optimization of Nitroxide-Based Inhibitors of Ferroptotic Cell Death in Cancer Cells and Macrophages
Author:
Affiliation:
1. Department of Chemistry, University of Pittsburgh, Pittsburgh, Pennsylvania 15260, United States
2. Pharmaceutical Sciences, Duquesne University School of Pharmacy, 415 Mellon Hall, Pittsburgh, Pennsylvania 15282, United States
Funder
U.S. Department of Defense
Defense Threat Reduction Agency
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Drug Discovery,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.1c00561
Reference32 articles.
1. Cell death pathways: intricate connections and disease implications
2. SnapShot: Ferroptosis
3. Regulation of Ferroptotic Cancer Cell Death by GPX4
4. Synthetic Lethal Screening Identifies Compounds Activating Iron-Dependent, Nonapoptotic Cell Death in Oncogenic-RAS-Harboring Cancer Cells
5. Selenium Utilization by GPX4 Is Required to Prevent Hydroperoxide-Induced Ferroptosis
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