Design and Synthesis of Oleanolic Acid Trimers to Enhance Inhibition of Influenza Virus Entry-Reference-Cited by-同舟云学术

Design and Synthesis of Oleanolic Acid Trimers to Enhance Inhibition of Influenza Virus Entry

Published:2021-11-02 Issue:11 Volume:12 Page:1759-1765
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Shao Liang¹^ORCID,Yang Fan¹,Su Yangqing¹,Li Weijia¹,Zhang Jihong¹,Xu Huan²,Huang Boxuan³,Sun Mengsi²,Mu Yu²,Zhang Yuan¹,Yu Fei¹⁴

Affiliation:

1. Medical School of Kunming University of Science and Technology, Kunming, Yunnan 650500, China

2. Institute of Chemical Biology, Shenzhen Bay Laboratories, Shenzhen, Guangdong 518132, China

3. Institute for Advanced Study, Shenzhen University, Shenzhen, Guangdong 518052, China

4. State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing 100191, China

Funder

National Natural Science Foundation of China

Open-Fund Program of the State Key Laboratory of Natural and Biomimetic Drugs

Yunnan Fundamental Research Projects

Shenzhen Bay laboratory start up fund

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.1c00374

Reference20 articles.

1. Structure–Property Relationship Studies of Influenza A Virus AM2-S31N Proton Channel Blockers

2. Influenza (Seasonal). World Health Organization, November 6, 2018.https://www.who.int/news-room/fact-sheets/detail/influenza-(seasonal) (accessed 2021-07-08).

3. A small-molecule fusion inhibitor of influenza virus is orally active in mice

4. Baloxavir: First Global Approval

5. Influenza (Flu), Antiviral Drugs and Related Information. U.S. Food and Drug Administration, October 26, 2020. https://www.fda.gov/drugs/information-drug-class/influenza-flu-antiviral-drugs-and-related-information (accessed 2021-07-08).

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