Optimization of Versatile Oxindoles as Selective PI3Kδ Inhibitors-Reference-Cited by-同舟云学术

Optimization of Versatile Oxindoles as Selective PI3Kδ Inhibitors

Published:2020-11-19 Issue:12 Volume:11 Page:2461-2469
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Methot Joey L.^ORCID,Achab Abdelghani,Christopher Matthew,Zhou Hua,McGowan Meredeth A.,Trotter B. Wesley,Fradera Xavier^ORCID,Lesburg Charles A.^ORCID,Goldenblatt Peter,Hill Armetta,Chen Dapeng,Otte Karin M.,Augustin Martin¹,Shah Sanjiv,Katz Jason D.

Affiliation:

1. Proteros Biostructures, Martinsried 82152, Germany

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.0c00441

Reference33 articles.

1. PI3K signalling in inflammation

2. PI3K inhibitors in inflammation, autoimmunity and cancer

3. Idelalisib: First-in-Class PI3K Delta Inhibitor for the Treatment of Chronic Lymphocytic Leukemia, Small Lymphocytic Leukemia, and Follicular Lymphoma

4. Management of adverse events associated with idelalisib treatment: expert panel opinion

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