Scaffold Repurposing of in-House Chemical Library toward the Identification of New Casein Kinase 1 δ Inhibitors
Author:
Affiliation:
1. Department of Pharmaceutical and Pharmacological Sciences, University of Padova, via Marzolo 5, 35131 Padova, Italy
2. Department of Chemical and Pharmaceutical Sciences, University of Trieste, Piazzale Europa,1 34127 Trieste, Italia
Funder
Ministero dell'Istruzione, dell'Universit? e della Ricerca
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Drug Discovery,Biochemistry
Link
http://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.0c00028
Reference28 articles.
1. The casein kinase 1 family: participation in multiple cellular processes in eukaryotes
2. The CK1 Family: Contribution to Cellular Stress Response and Its Role in Carcinogenesis
3. Crystallographic studies of casein kinase I δ: toward a structural understanding of auto-inhibition
4. Impaired CK1 Delta Activity Attenuates SV40-Induced Cellular Transformation In Vitro and Mouse Mammary Carcinogenesis In Vivo
5. CK1δ Kinase Activity Is Modulated by Chk1-Mediated Phosphorylation
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