Discovery of CDZ173 (Leniolisib), Representing a Structurally Novel Class of PI3K Delta-Selective Inhibitors
Author:
Affiliation:
1. Global Discovery Chemistry, ‡PK Sciences, §Chemical Biology and Therapeutics, and ∥Autoimmunity, Transplantation and Inflammation, Novartis Institutes for BioMedical Research, Novartis Campus, CH-4002 Basel, Switzerland
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Drug Discovery,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.7b00293
Reference27 articles.
1. The emerging mechanisms of isoform-specific PI3K signalling
2. Cutting Edge: Differential Roles for Phosphoinositide 3-Kinases, p110γ and p110δ, in Lymphocyte Chemotaxis and Homing
3. The PI3K pathway: clinical inhibition in chronic lymphocytic leukemia
4. Phosphoinositide 3-kinase inhibitor suppresses interleukin-17 expression in a murine asthma model
5. Selective role of PI3Kδ in neutrophil inflammatory responses
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