Molecular Determinants of Topoisomerase I Poisoning by Lamellarins: Comparison with Camptothecin and Structure−Activity Relationships-Reference-Cited by-同舟云学术

Molecular Determinants of Topoisomerase I Poisoning by Lamellarins: Comparison with Camptothecin and Structure−Activity Relationships

Published:2005-05-03 Issue:11 Volume:48 Page:3796-3807
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Marco Esther¹,Laine William¹,Tardy Christelle¹,Lansiaux Amélie¹,Iwao Masatomo¹,Ishibashi Fumito¹,Bailly Christian¹,Gago Federico¹

Affiliation:

1. Departamento de Farmacología, Universidad de Alcalá, E-28871 Madrid, Spain, INSERM U-524 and Laboratoire de Pharmacologie Antitumorale du Centre Oscar Lambret, IRCL, Place de Verdun, F-59045 Lille, France, and Faculty of Engineering and Faculty of Fisheries, Nagasaki University, Nagasaki 852-8521, Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049060w

Reference47 articles.

1. Camptothecin induces protein-linked DNA breaks via mammalian DNA topoisomerase I.

2. Camptothecin: current perspectives

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