Novel D3 Selective Dopaminergics Incorporating Enyne Units as Nonaromatic Catechol Bioisosteres: Synthesis, Bioactivity, and Mutagenesis Studies
Author:
Affiliation:
1. Department of Chemistry and Pharmacy, Emil Fischer Center, Friedrich Alexander University, Schuhstrasse 19, 91052 Erlangen, Germany
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm800895v
Reference45 articles.
1. Unis, A. S.; Roberson, M. D.; Hill, K.; Hamblin, M. W.; Dorsa, D. W.Differential localization of D2versus D3mRNA in midgestational human forebrain by in situ hybridizationSociety of Neuroscience Abstracts;Society of Neuroscience:Washington, DC,1995, Vol.21, p1620.
2. Neurochemical findings in the MPTP model of Parkinson's disease
3. Attenuation of 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine (MPTP) neurotoxicity by the novel selective dopamine D3-receptor partial agonist FAUC 329 predominantly in the nucleus accumbens of mice
4. Dopamine D3 receptor ligands—Recent advances in the control of subtype selectivity and intrinsic activity
Cited by 42 articles. 订阅此论文施引文献 订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献
1. Natural Product-Inspired Dopamine Receptor Ligands;Journal of Medicinal Chemistry;2024-07-22
2. Elucidating the chemical dynamics of the elementary reactions of the 1-propynyl radical (CH3CC; X2A1) with 2-methylpropene ((CH3)2CCH2; X1A1);Physical Chemistry Chemical Physics;2024
3. Palladium-Catalyzed Homo-Dimerization of Terminal Alkynes;Synthesis;2023-07-06
4. Dopamine Receptor Ligand Selectivity—An In Silico/In Vitro Insight;Biomedicines;2023-05-17
5. Approach to the specificity and selectivity between D2 and D3 receptors by mutagenesis and binding experiments part I: Expression and characterization of D2 and D3 receptor mutants;Protein Science;2022-11-16
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线，采集、加工和组织学术论文而形成的新型学术文献查询和分析系统，可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容，当前同舟云学术共收录了国内外主流学术期刊6万余种，收集的期刊论文及会议论文总量共计约1.5亿篇，并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询！咨询电话：010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3