Discovery of a 2,4-Disubstituted Pyrrolo[1,2-f][1,2,4]triazine Inhibitor (BMS-754807) of Insulin-like Growth Factor Receptor (IGF-1R) Kinase in Clinical Development-Reference-Cited by-同舟云学术

Discovery of a 2,4-Disubstituted Pyrrolo[1,2-f][1,2,4]triazine Inhibitor (BMS-754807) of Insulin-like Growth Factor Receptor (IGF-1R) Kinase in Clinical Development

Published:2009-09-24 Issue:23 Volume:52 Page:7360-7363
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Wittman Mark D.¹,Carboni Joan M.²,Yang Zheng³,Lee Francis Y.²,Antman Melissa⁴,Attar Ricardo²,Balimane Praveen³,Chang Chiehying⁵,Chen Cliff²,Discenza Lorell²,Frennesson David¹,Gottardis Marco M.²,Greer Ann²,Hurlburt Warren²,Johnson Walter¹,Langley David R.⁵,Li Aixin²,Li Jianqing⁶,Liu Peiying¹,Mastalerz Harold¹,Mathur Arvind⁶,Menard Krista²,Patel Karishma³,Sack John⁵,Sang Xiaopeng¹,Saulnier Mark¹,Smith Daniel⁶,Stefanski Kevin⁴,Trainor George¹,Velaparthi Upender¹,Zhang Guifen¹,Zimmermann Kurt¹,Vyas Dolatrai M.¹

Affiliation:

1. Discovery Chemistry

2. Oncology Drug Discovery

3. Metabolism and Pharmacokinetics

4. Pharmacuetics

5. Macromolecular Structure

6. Department of Chemical Synthesis

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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