(S)-(+)-4-[7-(2,2-Dimethyl-1-oxopro- poxy)-4-methyl-2-[4-[2-(1-piperidinyl)- ethoxy]phenyl]-2H-1-benzopyran-3-yl]- phenyl 2,2-Dimethylpropanoate (EM-800): A Highly Potent, Specific, and Orally Active Nonsteroidal Antiestrogen-Reference-Cited by-同舟云学术

(S)-(+)-4-[7-(2,2-Dimethyl-1-oxopro- poxy)-4-methyl-2-[4-[2-(1-piperidinyl)- ethoxy]phenyl]-2H-1-benzopyran-3-yl]- phenyl 2,2-Dimethylpropanoate (EM-800): A Highly Potent, Specific, and Orally Active Nonsteroidal Antiestrogen

Published:1997-07-01 Issue:14 Volume:40 Page:2117-2122
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Gauthier Sylvain¹,Caron Brigitte¹,Cloutier Julie¹,Dory Yves L.¹,Favre Alexandre¹,Larouche Denis¹,Mailhot Josée¹,Ouellet Carl¹,Schwerdtfeger Annette¹,Leblanc Gilles¹,Martel Céline¹,Simard Jacques¹,Mérand Yves¹,Bélanger Alain¹,Labrie Claude¹,Labrie Fernand¹

Affiliation:

1. Laboratory of Molecular Endocrinology, CHUL Research Centre, Le Centre Hospitalier Universitaire de Québec and Laval University, Québec, G1V 4G2, Canada

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm970095o

Reference42 articles.

1. Cancer statistics, 1997

2. Tamoxifen in advanced breast cancer

3. Estrogenic Regulation of Growth and Polypeptide Growth Factor Secretion in Human Breast Carcinoma

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