Imidazolopiperazines: Hit to Lead Optimization of New Antimalarial Agents-Reference-Cited by-同舟云学术

Imidazolopiperazines: Hit to Lead Optimization of New Antimalarial Agents

Published:2011-06-06 Issue:14 Volume:54 Page:5116-5130
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Wu Tao¹²³⁴⁵,Nagle Advait¹²³⁴⁵,Kuhen Kelli¹²³⁴⁵,Gagaring Kerstin¹²³⁴⁵,Borboa Rachel¹²³⁴⁵,Francek Caroline¹²³⁴⁵,Chen Zhong¹²³⁴⁵,Plouffe David¹²³⁴⁵,Goh Anne¹²³⁴⁵,Lakshminarayana Suresh B.¹²³⁴⁵,Wu Jeanette¹²³⁴⁵,Ang Hui Qing¹²³⁴⁵,Zeng Peiting¹²³⁴⁵,Kang Min Low¹²³⁴⁵,Tan William¹²³⁴⁵,Tan Maria¹²³⁴⁵,Ye Nicole¹²³⁴⁵,Lin Xuena¹²³⁴⁵,Caldwell Christopher¹²³⁴⁵,Ek Jared¹²³⁴⁵,Skolnik Suzanne¹²³⁴⁵,Liu Fenghua¹²³⁴⁵,Wang Jianling¹²³⁴⁵,Chang Jonathan¹²³⁴⁵,Li Chun¹²³⁴⁵,Hollenbeck Thomas¹²³⁴⁵,Tuntland Tove¹²³⁴⁵,Isbell John¹²³⁴⁵,Fischli Christoph¹²³⁴⁵,Brun Reto¹²³⁴⁵,Rottmann Matthias¹²³⁴⁵,Dartois Veronique¹²³⁴⁵,Keller Thomas¹²³⁴⁵,Diagana Thierry¹²³⁴⁵,Winzeler Elizabeth¹²³⁴⁵,Glynne Richard¹²³⁴⁵,Tully David C.¹²³⁴⁵,Chatterjee Arnab K.¹²³⁴⁵

Affiliation:

1. Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States

2. Swiss Tropical and Public Health Institute, Parasite Chemotherapy, Socinstrasse 57, Basel, Switzerland CH-4002

3. Novartis Institute for Tropical Diseases, 10 Biopolis Road, no. 05-01 Chromos, Singapore 138670

4. University of Basel, Petersplatz 1, Basel, Switzerland CH-4003

5. Novartis Institute for Biomedical Research, Preclinical Profiling Group, Cambridge, Massachusetts, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

http://pubs.acs.org/doi/pdf/10.1021/jm2003359

Reference32 articles.

1. Structure–activity relationships amongst 4-position quinoline methanol antimalarials that inhibit the growth of drug sensitive and resistant strains of Plasmodium falciparum

2. Anti-malarial activity of a non-piperidine library of next-generation quinoline methanols

3. A Research Agenda for Malaria Eradication: Drugs

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