Efficient Synthesis of 1,4-Thiazepanones and 1,4-Thiazepanes as 3D Fragments for Screening Libraries
Author:
Affiliation:
1. Department of Chemistry, University of Minnesota, Minneapolis, Minnesota 55455, United States
Funder
Masonic Cancer Center, University of Minnesota
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.orglett.0c01230
Reference30 articles.
1. Twenty years on: the impact of fragments on drug discovery
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