Stereoselective Synthesis of Either Exo- or Endo-3-Azabicyclo[3.1.0]hexane-6-carboxylates by Dirhodium(II)-Catalyzed Cyclopropanation with Ethyl Diazoacetate under Low Catalyst Loadings
Author:
Affiliation:
1. Department of Chemistry, Emory University, Atlanta, Georgia 30322, United States
2. Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, Indiana 46285, United States
Funder
Eli Lilly and Company
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.orglett.3c03652
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4. Synthesis and evaluation of 6-pyrazoylamido-3 N -substituted azabicyclo[3,1,0]hexane derivatives as T-type calcium channel inhibitors for treatment of neuropathic pain
5. Coates, D. A.; Remick, D. M. Preparation of novel SSTR4 agonist salts. WO2023044326, 2023.
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