Fast-Forwarding Hit to Lead: Aurora and Epidermal Growth Factor Receptor Kinase Inhibitor Lead Identification-Reference-Cited by-同舟云学术

Fast-Forwarding Hit to Lead: Aurora and Epidermal Growth Factor Receptor Kinase Inhibitor Lead Identification

Published:2010-06-15 Issue:13 Volume:53 Page:4980-4988
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Coumar Mohane Selvaraj¹,Chu Chang-Ying¹,Lin Cheng-Wei¹²,Shiao Hui-Yi¹,Ho Yun-Lung¹,Reddy Randheer¹,Lin Wen-Hsing¹,Chen Chun-Hwa¹,Peng Yi-Hui¹,Leou Jiun-Shyang¹,Lien Tzu-Wen¹,Huang Chin-Ting¹,Fang Ming-Yu¹,Wu Szu-Huei¹,Wu Jian-Sung¹,Chittimalla Santhosh Kumar¹,Song Jen-Shin¹,Hsu John T.-A.¹³,Wu Su-Ying¹,Liao Chun-Chen²⁴,Chao Yu-Sheng¹,Hsieh Hsing-Pang¹

Affiliation:

1. Division of Biotechnology and Pharmaceutical Research, National Health Research Institutes, 35 Keyan Road, Zhunan, Miaoli County 350, Taiwan, ROC

2. Department of Chemistry, National Tsing Hua University, 101 Guangfu Road Sec. 2, Hsinchu 300, Taiwan, ROC

3. Department of Biological Science and Technology, National Chiao Tung University, 1001 University Road, Hsinchu 300, Taiwan, ROC

4. Department of Chemistry, Chung Yuan Christian University, 200 Zhongbei Road, Zhongli 320, Taiwan, ROC

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm1000198

Reference26 articles.

1. FIGHTING THE CLOCK

2. Microtiter plate based chemistry and in situ screening: a useful approach for rapid inhibitor discovery

3. Protein Kinase Inhibitors: Insights into Drug Design from Structure

4. Roles of Aurora Kinases in Mitosis and Tumorigenesis

5. Aurora Kinases as Anticancer Drug Targets

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