Inhibitors of Ketohexokinase: Discovery of Pyrimidinopyrimidines with Specific Substitution that Complements the ATP-Binding Site-Reference-Cited by-同舟云学术

Inhibitors of Ketohexokinase: Discovery of Pyrimidinopyrimidines with Specific Substitution that Complements the ATP-Binding Site

Published:2011-04-28 Issue:7 Volume:2 Page:538-543
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Maryanoff Bruce E.¹,O'Neill John C.¹,McComsey David F.¹,Yabut Stephen C.¹,Luci Diane K.¹,Jordan Alfonzo D.¹,Masucci John A.¹,Jones William J.¹,Abad Marta C.¹,Gibbs Alan C.¹,Petrounia Ioanna¹

Affiliation:

1. Johnson & Johnson Pharmaceutical Research & Development, Spring House, Pennsylvania 19477-0776, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml200070g

Reference38 articles.

1. Fructose, insulin resistance, and metabolic dyslipidemia

2. Global and societal implications of the diabetes epidemic

3. The economic costs of NIDDM

4. Increased consumption of refined carbohydrates and the epidemic of type 2 diabetes in the United States: an ecologic assessment

5. Effects of dietary carbohydrates on glucose and lipid metabolism in golden Syrian hamsters

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