Fumaroylamino-4,5-epoxymorphinans and Related Opioids with Irreversible μ Opioid Receptor Antagonist Effects-Reference-Cited by-同舟云学术

Fumaroylamino-4,5-epoxymorphinans and Related Opioids with Irreversible μ Opioid Receptor Antagonist Effects

Published:2012-10-31 Issue:22 Volume:55 Page:9868-9874
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Moynihan Humphrey A.¹,Derrick Ian.¹,Broadbear Jillian H.²,Greedy Benjamin M.³,Aceto Mario D.⁴,Harris Louis S.⁴,Purington Lauren C. S.²,Thomas Mark P.³,Woods James H.²,Traynor John R.²,Husbands Stephen M.³,Lewis John W.³

Affiliation:

1. School of Chemistry, University of Bristol, Bristol, BS8 1TS, U.K.

2. Department of Pharmacology, University of Michigan, Michigan 48109, United States

3. Department of Pharmacy and Pharmacology, University of Bath, Bath, BA2 7AY, U.K.

4. Department of Pharmacology and Toxicology, Virginia Commonwealth University, Richmond, Virginia 23298, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm301096s

Reference25 articles.

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4. Cinnamoyl Derivatives of 7α-Aminomethyl-6,14-endo-ethanotetrahydrothebaine and 7α-Aminomethyl-6,14-endo-ethanotetrahydrooripavine and Related Opioid Ligands

5. Structural Determinants of Opioid Activity in Derivatives of 14-Aminomorphinones: Effect of Substitution in the Aromatic Ring of Cinnamoylaminomorphinones and Codeinones

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