Structure–Activity Relationship Study of Opiorphin, a Human Dual Ectopeptidase Inhibitor with Antinociceptive Properties-Reference-Cited by-同舟云学术

Structure–Activity Relationship Study of Opiorphin, a Human Dual Ectopeptidase Inhibitor with Antinociceptive Properties

Published:2012-01-25 Issue:3 Volume:55 Page:1181-1188
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Rosa Mònica¹,Arsequell Gemma¹,Rougeot Catherine²,Calle Luis P.³,Marcelo Filipa³,Pinto Marta⁴,Centeno Nuria B.⁴,Jiménez-Barbero Jesús³,Valencia Gregorio¹

Affiliation:

1. Institute of Advanced Chemistry of Catalonia (IQAC-CSIC), Barcelona, Spain

2. Institut Pasteur-Unité de Biochimie Structurale et Cellulaire/URA2185—CNRS, Paris, France

3. Chemical and Physical Biology, Centro de Investigaciones Biológicas (CIB-CSIC), Madrid, Spain

4. Computer-Assisted Drug Design Laboratory, Research Group on Biomedical Informatics (GRIB), IMIM-Universitat Pompeu Fabra, Barcelona, Spain

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm2012112

Reference46 articles.

1. Novel approaches to targeting neuropeptide systems

2. Protection of endogenous enkephalin catabolism as natural approach to novel analgesic and antidepressant drugs

3. Structure of human neutral endopeptidase (neprilysin) complexed with phosphoramidon 1 1Edited by R. Huber

4. Structural analysis of neprilysin with various specific and potent inhibitors

5. Structural studies of a bifunctional inhibitor of neprilysin and DPP-IV

Cited by 16 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Opiorphin: an endogenous human peptide with intriguing application in diverse range of pathologies;Inflammopharmacology;2024-08-20

2. Time-course of pain and salivary opiorphin release in response to oral capsaicin differ in burning mouth syndrome patients, temporomandibular disorders patients and control subjects;Clinical Oral Investigations;2024-04-09

3. Enhancing Opiorphin’s Metabolic Stability and Preserving its Potent Analgesic Effect: A Systematic Review;Current Topics in Medicinal Chemistry;2024-01

4. Harnessing conformational drivers in drug design;Progress in Medicinal Chemistry;2024

5. A possible alternative to Opiorphin and its stable analogues for treating fibromyalgia pain: A clinical hypothesis;Northern Clinics of Istanbul;2022