Structure-Based Design of Potent and Ligand-Efficient Inhibitors of CTX-M Class A β-Lactamase-Reference-Cited by-同舟云学术

Structure-Based Design of Potent and Ligand-Efficient Inhibitors of CTX-M Class A β-Lactamase

Published:2012-02-14 Issue:5 Volume:55 Page:2163-2172
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Nichols Derek A.¹,Jaishankar Priyadarshini²,Larson Wayne²,Smith Emmanuel¹,Liu Guoqing¹,Beyrouthy Racha³,Bonnet Richard³,Renslo Adam R.²,Chen Yu¹

Affiliation:

1. University of South Florida College of Medicine, Department of Molecular Medicine,12901 Bruce B. Downs Boulevard, MDC 3522, Tampa, Florida 33612, United States

2. Department of Pharmaceutical Chemistry and Small Molecule Discovery Center, University of California San Francisco, 1700 Fourth Street, Byers Hall S504, San Francisco, California 94158, United States

3. Clermont Université, Université d’Auvergne, M2iSH, BP10448, INRA, USC 2018, CHU Clermont-Ferrand, Service de Bactériologie, F-63003 Clermont-Ferrand, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm2014138

Reference43 articles.

1. Crystal Structures of Penicillin-Binding Protein 6 from Escherichia coli

2. The future of the β-lactams

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4. The Crystal Structure of Phosphonate-Inhibited d-Ala-d-Ala Peptidase Reveals an Analogue of a Tetrahedral Transition State,

5. Beta-lactamases and bacterial resistance to antibiotics

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