Bisubstrate inhibitors: the promise of a selective and potent chemical inhibition of epigenetic ‘writers’-Reference-Cited by-同舟云学术

Bisubstrate inhibitors: the promise of a selective and potent chemical inhibition of epigenetic ‘writers’

Published:2020-09 Issue:17 Volume:12 Page:1479-1482
ISSN:1750-1911
Container-title:Epigenomics
language:en
Short-container-title:Epigenomics

Author:

Bon Corentin¹^ORCID,Halby Ludovic¹^ORCID,Arimondo Paola Barbara¹^ORCID

Affiliation:

1. Department of Structural Biology & Chemistry, EpiCBio, Epigenetic Chemical Biology, Institut Pasteur, CNRS UMR n°3523, 28 rue du Dr Roux, 75015 Paris, France

Publisher

Future Medicine Ltd

Subject

Cancer Research,Genetics

Link

https://www.futuremedicine.com/doi/pdf/10.2217/epi-2020-0203

Reference19 articles.

1. Selective Inhibition of EZH2 by EPZ-6438 Leads to Potent Antitumor Activity in EZH2-Mutant Non-Hodgkin Lymphoma

2. SAM/SAH Analogs as Versatile Tools for SAM-Dependent Methyltransferases

3. Structural Chemistry of the Histone Methyltransferases Cofactor Binding Site

4. SET domain protein lysine methyltransferases: Structure, specificity and catalysis

5. Structural Biology of Human H3K9 Methyltransferases

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4. Bisubstrate Strategies to Target Methyltransferases;European Journal of Organic Chemistry;2022-02-21

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