1. Modified peptides are being defined as peptides in which in essence the amino acid sequence is unchanged but the peptide contains e. g. some unnatural amino acids a modification of a cysteine residue or a phospho amino acid.Peptidomimeticsare compounds which imitate the structure and/or imitate or block the biological effect of a peptide at the receptor level [2a]. As a consequence peptidomimetics span the whole range of compounds varying from peptide isosteres to compounds without an identifiable amino acid or peptide moiety.
2. Peptidomimetics for Receptor Ligands?Discovery, Development, and Medical Perspectives
3. Conformationally restricted amino acids and dipeptides, (non)peptidomimetics and secondary structure mimetics
4. Case histories of peptidomimetics: Progression from peptides to drugs
5. Peptidomimetics—Tailored Enzyme Inhibitors