Structure‐Based Design of FXIIIa‐Blockers: Addressing a Transient Hydrophobic Pocket in the Active Site of FXIIIa-Reference-Cited by-同舟云学术

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Structure‐Based Design of FXIIIa‐Blockers: Addressing a Transient Hydrophobic Pocket in the Active Site of FXIIIa

Published:2020-04-07 Issue:10 Volume:15 Page:900-905
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Stieler Martin¹,Büchold Christian²,Schmitt Marisa²,Heine Andreas¹^ORCID,Hils Martin²,Pasternack Ralf²,Klebe Gerhard¹^ORCID

Affiliation:

1. Department of Pharmaceutical ChemistryPhilipps-Universität Marbacher Weg 6 35032 Marburg Germany

2. Zedira GmbH Roesslerstrasse 83 64293 Darmstadt Germany

Funder

Helmholtz-Zentrum Berlin für Materialien und Energie

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/cmdc.202000056

Reference38 articles.

1. Transglutaminases: crosslinking enzymes with pleiotropic functions

2. Protein Crosslinking in Assembly and Remodelling of Extracellular Matrices: The Role of Transglutaminases

3. Expression of Transglutaminase 1 in Human Epidermis

4. Transglutaminase 5 Cross-links Loricrin, Involucrin, and Small Proline-rich Proteins in Vitro

5. Expression of Transglutaminase 5 in Normal and Pathologic Human Epidermis

Cited by 3 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Discovery of Heparin Mimetic, Potent, and Selective Inhibitors of Human Clotting Factor XIIIa;ACS Omega;2024-07-03

2. Autoantibody binding and unique enzyme-substrate intermediate conformation of human transglutaminase 3;Nature Communications;2023-10-05

3. Peptidic Inhibitors and a Fluorescent Probe for the Selective Inhibition and Labelling of Factor XIIIa Transglutaminase;Molecules;2023-02-08

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